PAPOT Sebastien

Sebastien PAPOT

Professor Sênior – Université de Poitiers

Equipe: Síntese Orgânica

Palavras-chave: chimiothérapie anticancéreuse, vectorização thérapeutique, prodrogue, nanosystème, chimie prébiotique

Contato

IC2MP
Equipe «Synthèse»
Anexo bâtiment B27
Université de Poitiers de
4 rue Michel Brunet
86022 Poitiers
tel: (+) 33 (0) 5 49 45 38 62

e-mail: sebastien.papot[at]univ-poitiers.fr

Publicações importantes:

– Efficient regio and stereoselective Synthesis of 1-b-O-Glucuronyl Carbamates and Carbonates from 1,2,3,4-Hydroxyl Unprotected Glucuronates.
M. Thomas, J.-P. Gesson and S. Papot Synlett 2007, 12, 1966-1968.

– First O-Glycosylation of Hydroxamic Acids.
M. Thomas, J.-P. Gesson and S. Papot
The Journal of Organic Chemistry 2007, 72, 4262-4264.

– Synthesis and Biological Evaluation of the Suberoylanilide Hydroxamic Acid (SAHA) b-glucuronide and b-galactoside for Application in Selective Prodrug Chemotherapy.
M. Thomas, Freddy Rivault, Isabelle Tranoy-Opalinski, Joëlle Roche, Jean-Pierre Gesson and Sébastien Papot
Bioorganic and Medicinal Chemistry Letters 2007, 17, 983-986.

– A New Simple and Convenient Method for the Synthesis of Substituted 2,6,9-Trioxabicyclo[3.3.1]-nona-3,7-dienes from Arylmalondialdehydes.
A. Fernandes, J. Marrot, J.P. Gesson, S. Papot
Tetrahedron Lett. 2006, 47. 5961-5964.

– Looking Forward: A Glance into the Future of Organic Chemistry.
P. COMPAIN, V. DESVERGNES, C. OLLIVIER, F. ROBERT, F. SUZENET, M. BARBOIU, P. BELMONT, Y. BLERIOT, F. BOLZE, S. BOUQUILLON, E. BOURGUET, B. BRAIDA, T. CONSTANTIEUX, L. DESAUBRY, D. DUPONT, S. GASTALDI, F. JEROME, S. LEGOUPY, X. MARAT, M. MIGAUD, N. MOITESSIER, S. PAPOT, F. PERI, M. PETIT, S. PY, E. SCHULZ, I. TRANOY-OPALINSKI, B. VAUZEILLES, P. VAYRON, L. VERGNES, S. VIDAL, S. WILMOUTH.
New J. Chem. 2006, 30, 823-831.

– Design of Selectively Activated Anticancer Prodrugs: Elimination and Cyclisation Strategies (review)
S. PAPOT, I. TRANOY, F. TILLEQUIN, J-C. FLORENT, J-P. GESSON
Curr. Med. Chem.-Anti-Cancer Agents 2002, 2, 155-185.

– Synthesis of Indomethacin Analogues for Evaluation as Moderators of MRP
A.R. MAGUIRE, S.J. PLUNKETT, S. PAPOT, M. CLYNES, R. O’CONNOR, S. TOUHEY
Bioorg. Med. Chem. 2001, 9, 745-762.

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